The obtained BCP sulfides were oxidized and iminated to obtain BCP sulfoxides and sulfoximines. These modifications to tune parameters like the polarity are important for a successful application of the structural motif in drug design. The final aim of this thesis was the synthesis and application of a bench-stable BCP building block to facilitate the use in medicinal chemistry and other fields. A facile and scalable four-step route to sodium BCP sulfinate was developed to deliver the product in good yield and purity. The sulfinate was applied in the synthesis of BCP sulfones, sulfoxides, a sulfinamide and sulfonamides.
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